Bulk Kisspeptin-10
kisspeptin receptor and neuroendocrine signaling research research material, supplied as a lyophilized reference standard. >=99% by HPLC.
Available Sizes & Pricing
| Size | Price per vial (USD) |
|---|---|
| 5 mg | $64.95 |
| 10 mg | $99.95 |
A minimum inquiry quantity of 10 vials applies across requested products. Inquire for bulk purchase or larger lot quantities →
Bulk Kisspeptin-10 Specifications
| CAS Number | See lot-specific COA |
|---|---|
| Molecular Formula | See lot-specific COA |
| Molecular Weight | See lot-specific COA |
| Purity | >=99% by HPLC |
| Storage | Store lyophilized material at -20 C. Avoid repeated freeze-thaw cycles after reconstitution. |
What Is Kisspeptin-10?
Kisspeptin-10 is cataloged for controlled laboratory workflows focused on kisspeptin receptor and neuroendocrine signaling research. Its lot-specific analytical documentation should be reviewed alongside the receiving laboratory's established handling and assay-validation procedures. For laboratory research use only - not for human or veterinary use.
Kisspeptin-10 Research Context
Kisspeptin-10 (KP-10; KISS1 protein 45-54) is the C-terminal decapeptide fragment of the kisspeptin family and the minimal active sequence for KISS1R (GPR54) activation. It is a primary reference tool compound for studying KISS1R-dependent Gq/11 signaling and intracellular calcium mobilization in neuroendocrine cell models. Because KISS1R is expressed in GnRH neurons, KP-10 is used in hypothalamic cell research examining upstream neuroendocrine signaling cascades.
KP-10 binds KISS1R and activates Gq/11-coupled phospholipase C-β, generating IP₃ and DAG, which release intracellular Ca²⁺ from ER stores. This calcium signal is measured by fluorescent calcium dyes (Fluo-4, Fura-2) in real-time FLIPR-format assays in KISS1R-transfected HEK293 or neuroendocrine cell lines.
Study-Design Considerations
- Calcium-flux assays with KP-10 require rapid compound addition (≤5 s lag) and pre-loading cells with the calcium indicator 45–60 min before the assay; sub-optimal dye loading conditions produce underestimated EC₅₀ values.
- Include a KISS1R-negative cell line as a specificity control to confirm that calcium responses are receptor-mediated rather than non-specific peptide-induced membrane permeabilization.
Interpretation Limits
KISS1R calcium signals in transfected non-neuroendocrine lines do not model the complex GnRH-neuron context in which endogenous kisspeptin signaling is physiologically relevant.
Kisspeptin-10 Research Applications
- KISS1R receptor assays
- Neuroendocrine signaling
- Ligand-binding studies
Source Records
Use the following scientific and compound-record sources when developing a laboratory-specific protocol; they do not replace method validation for a particular lot or assay.
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Buy Bulk Kisspeptin-10 for Research
Bulk Peptides supplies bulk Kisspeptin-10 to institutional laboratories, CROs, and research facilities across the United States. Every lot is characterized by reverse-phase HPLC at 220 nm and confirmed by electrospray ionization mass spectrometry before shipping. A lot-specific Certificate of Analysis documents both results for your records.
Bulk Kisspeptin-10 is available in the catalog sizes above. A minimum inquiry quantity of 10 vials applies; contact us for larger requirements or custom synthesis quotes. All products are for laboratory research use only (RUO) — not for human or veterinary use.
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